Well | KIT 1 | KIT 2 |
compound | 結果 | compound | 結果 |
1 -
A | none (DMSO) | 100.0
| none (DMSO) | 100.0
|
1 -
B | 5-FU | 78.6
| Pifithrin-a (cyclic) | 99.8
|
1 -
C | Bestatin Hydrochloride | 128.4
| PRIMA-1 | 103.5
|
1 -
D | Bleomycin sulfate | 78.8
| Finasteride | 108.6
|
1 -
E | Cisplatin | 109.6
| Aminoglutethimide | 98.6
|
1 -
F | Methotrexate | 54.7
| Formestane | 114.9
|
1 -
G | Mitomycin C | 10.4
| Mifepristone | 101.6
|
1 -
H | Vinblastine sulfate | 5.3
| TOFA | 134.7
|
2 -
A | Paclitaxel | 69.6
| Amastatin | 111.9
|
2 -
B | Flutamide | 104.6
| Actinonin | 87.4
|
2 -
C | Daunorubicin, HCl | 24.3
| Oligomycin | -0.2
|
2 -
D | Doxorubicin, HCl | 41.2
| Bafilomycin A1 | 0.2
|
2 -
E | Tamoxifen, citrate | 8.9
| HA 14-1 | 100.5
|
2 -
F | Actinomycin D | 33.3
| BH3I-1 | 97.9
|
2 -
G | Camptothecin | 6.0
| LFM-A13 | 118.6
|
2 -
H | Aclarubicin | 22.7
| Terreic acid | 122.3
|
3 -
A | Etoposide (VP-16) | 23.4
| E-64d | 118.6
|
3 -
B | Cytochalasin D | 53.5
| ALLN | 7.9
|
3 -
C | 2',5'-dideoxyadenosine | 116.4
| CA-074 | 100.0
|
3 -
D | AKT inhibitor | 121.2
| Pepstatin A | 100.0
|
3 -
E | NL-71-101 | 128.0
| Z-GLF-CMK | 95.1
|
3 -
F | AG957 | 112.3
| RS 102895 | 110.2
|
3 -
G | KN93 | 106.5
| SB 328437 | 106.0
|
3 -
H | Z-VAD-FMK | 119.0
| SB 225002 | 41.2
|
4 -
A | Kenpaullone | 93.3
| AMD3100 octahydrochloride | 116.7
|
4 -
B | Purvalanol A | 76.6
| NSC95397 | 121.6
|
4 -
C | 3-ATA | 95.2
| SC-ααδ9 | 96.3
|
4 -
D | Olomoucine | 92.8
| Amiloride | 94.7
|
4 -
E | TBB | 94.2
| Lidocaine | 89.1
|
4 -
F | Sulindac sulfide | 92.8
| Monensin | 14.9
|
4 -
G | Valeryl salicylate | 96.1
| Ouabain | 14.9
|
4 -
H | NS-398 | 110.8
| Sanguinarine | -1.9
|
5 -
A | Sodium salicylate | 116.6
| Glibenclamide | 112.1
|
5 -
B | Theophylline | 107.7
| Dequalinium | 29.3
|
5 -
C | Azacytidine | 6.7
| Diazoxide | 95.1
|
5 -
D | Aphidicolin | 74.0
| Valinomycin | 5.6
|
5 -
E | AG1478 | 80.5
| Nigericin | 8.8
|
5 -
F | Genistein | 108.2
| Diltiazem | 101.2
|
5 -
G | Manumycin A | 130.8
| Nifedipine | 90.5
|
5 -
H | FTI-276 | 108.4
| Verapamil | 88.1
|
6 -
A | SU1498 | 90.6
| PGP-4008 | 119.8
|
6 -
B | GGTI-286 | 102.7
| Fumitremorgin C | 90.7
|
6 -
C | Dexamethasone | 92.0
| A23187 | 2.3
|
6 -
D | GSK-3 inhibitor II | 112.5
| Ionomycin | 5.3
|
6 -
E | Scriptaid | 14.5
| Thapsigargin | 8.4
|
6 -
F | Trichostatin A | 16.4
| t-Butylhydroquinone (BHQ) | 114.0
|
6 -
G | AG825 | 101.7
| N-phenylanthranilic acid | 107.9
|
6 -
H | Cycloheximide | 51.6
| DIDS | 117.4
|
7 -
A | Lovastatin | 93.7
| SB 218078 | 50.9
|
7 -
B | Radicicol | 49.9
| Debromohymenialdisine (DBH) | 92.3
|
7 -
C | 17-AAG | 53.5
| Rotenone | 35.6
|
7 -
D | AG1024 | 101.9
| Antimycin A1 | 102.8
|
7 -
E | 1400W, HCl | 105.1
| Leptomycin B* | 21.2
|
7 -
F | AMT, HCl | 103.1
| R59022 | 103.7
|
7 -
G | AG490 | 126.5
| Dioctanoylglycol | 107.0
|
7 -
H | Cucurbitacin I | 6.3
| RHC80267 | 99.5
|
8 -
A | SP600125 | 51.6
| Xanthohumol | 80.9
|
8 -
B | Damnacanthal | 123.1
| C75 | 99.5
|
8 -
C | PD 98059 | 130.8
| Cerulenin | 99.8
|
8 -
D | U0126 | 88.2
| Tunicamycin | 27.9
|
8 -
E | Fumagillin | 114.7
| Deoxynojirimycin | 92.6
|
8 -
F | GM 6001 | 102.4
| Swainsonine | 97.9
|
8 -
G | N-Acetyl-L-cysteine | 114.7
| LY 83583 | 17.4
|
8 -
H | Aminoguanidine, HCl | 129.4
| ODQ | 70.2
|
9 -
A | L-NMMA | 123.9
| Anacardic acid | 110.9
|
9 -
B | PD169316 | 110.6
| Chetomin | 21.6
|
9 -
C | SB 203580 | 98.8
| Dimethyloxalylglycine | 94.0
|
9 -
D | Rapamycin | 74.7
| HR22C16 | 67.0
|
9 -
E | NU1025 | 106.3
| Monastrol | 92.8
|
9 -
F | Benzamide | 114.0
| Nordihydroguaiaretic acid (NDGA) | 108.8
|
9 -
G | D609 | 117.8
| ETYA | 123.0
|
9 -
H | IBMX | 106.0
| Baicalein | 86.0
|
10 -
A | Ro-20-1724 | 133.3
| Nutlin-3 | 101.6
|
10 -
B | Zaprinast | 95.7
| MDM2 inhibitor | 97.7
|
10 -
C | AG1296 | 99.3
| Phenelzine | 93.7
|
10 -
D | LY294002 | 64.8
| Deprenyl | 105.8
|
10 -
E | Wortmannin | 89.6
| Decylubiquinone | 106.7
|
10 -
F | H-89, HCl | 89.2
| Ro 5-4864 | 94.4
|
10 -
G | Bisindolymaleimide I, HCl | 53.0
| Lonidamine | 101.6
|
10 -
H | H-7 | 141.9
| ML-7 | 84.4
|
11 -
A | Staurosporine | 7.7
| Benzylguanine | 96.0
|
11 -
B | cPLA2inhibitor | 107.5
| DFMO | 113.0
|
11 -
C | OBAA | 103.6
| KT 5823 | 67.9
|
11 -
D | Cantharidin | 9.9
| Rp-8-CPT-cGMPS | 109.3
|
11 -
E | Cytostatin | 22.9
| MK 886 | 106.0
|
11 -
F | Cyclosporin A | 16.9
| Clofibrate | 116.5
|
11 -
G | FK-506 | 133.5
| BADGE | 105.6
|
11 -
H | MG-132 | 3.9
| Troglitazone | 102.3
|
12 -
A | Lactacystin | 145.3
| AZT | 118.8
|
12 -
B | Hydroxyurea | 124.8
| Nalidixic acid | 102.1
|
12 -
C | HA1077 | 98.3
| a-Amanitin | 52.6
|
12 -
D | Y27632 | 97.1
| MST-312 | 79.1
|
12 -
E | PP1 (analog) | 118.6
| b-Rubromycin | 25.3
|
12 -
F | PP-H | 126.3
| SB 431542 | 135.1
|
12 -
G | Nocodazole | 29.9
| N1,N12-Diethylspermine (BESpm) | 117.0
|
12 -
H | Dephostatin | 107.5
| Fumonisin B1 | 121.4
|