Well | KIT 1 | KIT 2 |
compound | 結果 | compound | 結果 |
1 -
A | none (DMSO) | 100.0
| none (DMSO) | 100.0
|
1 -
B | 5-FU | 78.3
| Pifithrin-a (cyclic) | 86.6
|
1 -
C | Bestatin Hydrochloride | 92.6
| PRIMA-1 | 91.8
|
1 -
D | Bleomycin sulfate | 70.2
| Finasteride | 97.0
|
1 -
E | Cisplatin | 91.9
| Aminoglutethimide | 93.1
|
1 -
F | Methotrexate | 65.9
| Formestane | 104.3
|
1 -
G | Mitomycin C | 24.4
| Mifepristone | 82.8
|
1 -
H | Vinblastine sulfate | 38.0
| TOFA | 105.6
|
2 -
A | Paclitaxel | 59.3
| Amastatin | 94.8
|
2 -
B | Flutamide | 82.2
| Actinonin | 92.7
|
2 -
C | Daunorubicin, HCl | 12.8
| Oligomycin | 6.9
|
2 -
D | Doxorubicin, HCl | 4.7
| Bafilomycin A1 | -1.3
|
2 -
E | Tamoxifen, citrate | 8.9
| HA 14-1 | 90.9
|
2 -
F | Actinomycin D | 26.0
| BH3I-1 | 94.0
|
2 -
G | Camptothecin | -2.3
| LFM-A13 | 96.6
|
2 -
H | Aclarubicin | 10.9
| Terreic acid | 68.5
|
3 -
A | Etoposide (VP-16) | 31.4
| E-64d | 131.9
|
3 -
B | Cytochalasin D | 46.5
| ALLN | 27.2
|
3 -
C | 2',5'-dideoxyadenosine | 94.2
| CA-074 | 100.9
|
3 -
D | AKT inhibitor | 108.9
| Pepstatin A | 97.0
|
3 -
E | NL-71-101 | 96.1
| Z-GLF-CMK | 67.7
|
3 -
F | AG957 | 97.7
| RS 102895 | 106.0
|
3 -
G | KN93 | 81.8
| SB 328437 | 111.2
|
3 -
H | Z-VAD-FMK | 105.4
| SB 225002 | 65.9
|
4 -
A | Kenpaullone | 36.0
| AMD3100 octahydrochloride | 113.8
|
4 -
B | Purvalanol A | 44.6
| NSC95397 | 126.7
|
4 -
C | 3-ATA | 85.7
| SC-ααδ9 | 115.1
|
4 -
D | Olomoucine | 84.9
| Amiloride | 91.8
|
4 -
E | TBB | 78.7
| Lidocaine | 88.4
|
4 -
F | Sulindac sulfide | 82.9
| Monensin | 38.4
|
4 -
G | Valeryl salicylate | 82.6
| Ouabain | 10.3
|
4 -
H | NS-398 | 100.0
| Sanguinarine | -5.2
|
5 -
A | Sodium salicylate | 98.4
| Glibenclamide | 106.9
|
5 -
B | Theophylline | 82.2
| Dequalinium | 75.0
|
5 -
C | Azacytidine | 3.1
| Diazoxide | 106.9
|
5 -
D | Aphidicolin | 39.5
| Valinomycin | 12.1
|
5 -
E | AG1478 | 69.4
| Nigericin | 23.7
|
5 -
F | Genistein | 83.7
| Diltiazem | 105.6
|
5 -
G | Manumycin A | 88.8
| Nifedipine | 99.1
|
5 -
H | FTI-276 | 89.9
| Verapamil | 89.2
|
6 -
A | SU1498 | 13.2
| PGP-4008 | 111.6
|
6 -
B | GGTI-286 | 84.9
| Fumitremorgin C | 104.7
|
6 -
C | Dexamethasone | 84.1
| A23187 | 4.7
|
6 -
D | GSK-3 inhibitor II | 86.4
| Ionomycin | 11.2
|
6 -
E | Scriptaid | 6.2
| Thapsigargin | 18.1
|
6 -
F | Trichostatin A | 8.9
| t-Butylhydroquinone (BHQ) | 56.5
|
6 -
G | AG825 | 83.3
| N-phenylanthranilic acid | 95.7
|
6 -
H | Cycloheximide | 24.0
| DIDS | 100.0
|
7 -
A | Lovastatin | 92.2
| SB 218078 | 41.8
|
7 -
B | Radicicol | 50.4
| Debromohymenialdisine (DBH) | 96.1
|
7 -
C | 17-AAG | 48.4
| Rotenone | 68.5
|
7 -
D | AG1024 | 122.1
| Antimycin A1 | 97.0
|
7 -
E | 1400W, HCl | 83.3
| Leptomycin B* | 35.8
|
7 -
F | AMT, HCl | 83.7
| R59022 | 103.4
|
7 -
G | AG490 | 93.4
| Dioctanoylglycol | 131.0
|
7 -
H | Cucurbitacin I | 5.8
| RHC80267 | 96.6
|
8 -
A | SP600125 | 65.5
| Xanthohumol | 96.6
|
8 -
B | Damnacanthal | 93.8
| C75 | 113.4
|
8 -
C | PD 98059 | 96.9
| Cerulenin | 116.4
|
8 -
D | U0126 | 89.9
| Tunicamycin | 18.1
|
8 -
E | Fumagillin | 84.9
| Deoxynojirimycin | 94.4
|
8 -
F | GM 6001 | 94.2
| Swainsonine | 100.4
|
8 -
G | N-Acetyl-L-cysteine | 97.7
| LY 83583 | 22.0
|
8 -
H | Aminoguanidine, HCl | 90.7
| ODQ | 83.2
|
9 -
A | L-NMMA | 105.8
| Anacardic acid | 108.6
|
9 -
B | PD169316 | 86.8
| Chetomin | 22.4
|
9 -
C | SB 203580 | 93.4
| Dimethyloxalylglycine | 97.4
|
9 -
D | Rapamycin | 69.4
| HR22C16 | 78.9
|
9 -
E | NU1025 | 95.7
| Monastrol | 105.2
|
9 -
F | Benzamide | 88.8
| Nordihydroguaiaretic acid (NDGA) | 111.2
|
9 -
G | D609 | 102.7
| ETYA | 106.0
|
9 -
H | IBMX | 90.7
| Baicalein | 90.1
|
10 -
A | Ro-20-1724 | 108.9
| Nutlin-3 | 104.7
|
10 -
B | Zaprinast | 79.8
| MDM2 inhibitor | 76.7
|
10 -
C | AG1296 | 69.4
| Phenelzine | 119.4
|
10 -
D | LY294002 | 75.2
| Deprenyl | 109.1
|
10 -
E | Wortmannin | 79.1
| Decylubiquinone | 116.8
|
10 -
F | H-89, HCl | 77.5
| Ro 5-4864 | 109.9
|
10 -
G | Bisindolymaleimide I, HCl | 36.0
| Lonidamine | 111.2
|
10 -
H | H-7 | 104.7
| ML-7 | 89.7
|
11 -
A | Staurosporine | 8.1
| Benzylguanine | 126.3
|
11 -
B | cPLA2inhibitor | 93.4
| DFMO | 115.1
|
11 -
C | OBAA | 80.6
| KT 5823 | 81.9
|
11 -
D | Cantharidin | 27.1
| Rp-8-CPT-cGMPS | 107.8
|
11 -
E | Cytostatin | 38.8
| MK 886 | 103.0
|
11 -
F | Cyclosporin A | 17.8
| Clofibrate | 130.2
|
11 -
G | FK-506 | 100.4
| BADGE | 100.9
|
11 -
H | MG-132 | 3.9
| Troglitazone | 101.3
|
12 -
A | Lactacystin | 114.7
| AZT | 121.1
|
12 -
B | Hydroxyurea | 103.9
| Nalidixic acid | 119.0
|
12 -
C | HA1077 | 108.9
| a-Amanitin | 47.0
|
12 -
D | Y27632 | 111.2
| MST-312 | 21.1
|
12 -
E | PP1 (analog) | 105.0
| b-Rubromycin | 65.1
|
12 -
F | PP-H | 111.2
| SB 431542 | 146.6
|
12 -
G | Nocodazole | 63.6
| N1,N12-Diethylspermine (BESpm) | 110.3
|
12 -
H | Dephostatin | 99.2
| Fumonisin B1 | 75.9
|