Well | KIT 1 | KIT 2 |
compound | 結果 | compound | 結果 |
1 -
A | none (DMSO) | 100.0
| none (DMSO) | 100.0
|
1 -
B | 5-FU | 75.3
| Pifithrin-a (cyclic) | 88.8
|
1 -
C | Bestatin Hydrochloride | 102.8
| PRIMA-1 | 99.7
|
1 -
D | Bleomycin sulfate | 100.7
| Finasteride | 110.0
|
1 -
E | Cisplatin | 96.0
| Aminoglutethimide | 99.6
|
1 -
F | Methotrexate | 59.6
| Formestane | 99.5
|
1 -
G | Mitomycin C | 47.9
| Mifepristone | 87.3
|
1 -
H | Vinblastine sulfate | 33.9
| TOFA | 55.4
|
2 -
A | Paclitaxel | 49.2
| Amastatin | 88.2
|
2 -
B | Flutamide | 80.8
| Actinonin | 66.9
|
2 -
C | Daunorubicin, HCl | 26.9
| Oligomycin | 36.5
|
2 -
D | Doxorubicin, HCl | 32.9
| Bafilomycin A1 | 14.1
|
2 -
E | Tamoxifen, citrate | 27.2
| HA 14-1 | 85.1
|
2 -
F | Actinomycin D | 25.8
| BH3I-1 | 94.4
|
2 -
G | Camptothecin | 33.8
| LFM-A13 | 82.2
|
2 -
H | Aclarubicin | 21.1
| Terreic acid | 76.0
|
3 -
A | Etoposide (VP-16) | 67.9
| E-64d | 97.7
|
3 -
B | Cytochalasin D | 84.6
| ALLN | 62.6
|
3 -
C | 2',5'-dideoxyadenosine | 84.7
| CA-074 | 95.1
|
3 -
D | AKT inhibitor | 100.4
| Pepstatin A | 88.7
|
3 -
E | NL-71-101 | 96.5
| Z-GLF-CMK | 97.8
|
3 -
F | AG957 | 91.3
| RS 102895 | 65.8
|
3 -
G | KN93 | 64.6
| SB 328437 | 91.2
|
3 -
H | Z-VAD-FMK | 99.4
| SB 225002 | 43.6
|
4 -
A | Kenpaullone | 68.9
| AMD3100 octahydrochloride | 118.8
|
4 -
B | Purvalanol A | 52.2
| NSC95397 | 125.0
|
4 -
C | 3-ATA | 88.2
| SC-ααδ9 | 81.9
|
4 -
D | Olomoucine | 94.4
| Amiloride | 95.0
|
4 -
E | TBB | 79.3
| Lidocaine | 79.6
|
4 -
F | Sulindac sulfide | 78.9
| Monensin | 45.3
|
4 -
G | Valeryl salicylate | 102.5
| Ouabain | 23.7
|
4 -
H | NS-398 | 86.8
| Sanguinarine | -1.5
|
5 -
A | Sodium salicylate | 99.0
| Glibenclamide | 88.5
|
5 -
B | Theophylline | 91.1
| Dequalinium | 42.8
|
5 -
C | Azacytidine | 49.9
| Diazoxide | 88.3
|
5 -
D | Aphidicolin | 85.0
| Valinomycin | 21.2
|
5 -
E | AG1478 | 66.3
| Nigericin | 26.2
|
5 -
F | Genistein | 80.0
| Diltiazem | 85.6
|
5 -
G | Manumycin A | 106.0
| Nifedipine | 76.8
|
5 -
H | FTI-276 | 94.2
| Verapamil | 77.9
|
6 -
A | SU1498 | 57.8
| PGP-4008 | 82.3
|
6 -
B | GGTI-286 | 87.1
| Fumitremorgin C | 81.0
|
6 -
C | Dexamethasone | 90.8
| A23187 | 2.8
|
6 -
D | GSK-3 inhibitor II | 75.8
| Ionomycin | 2.7
|
6 -
E | Scriptaid | 25.1
| Thapsigargin | 34.1
|
6 -
F | Trichostatin A | 26.4
| t-Butylhydroquinone (BHQ) | 91.7
|
6 -
G | AG825 | 78.3
| N-phenylanthranilic acid | 84.0
|
6 -
H | Cycloheximide | 46.8
| DIDS | 84.2
|
7 -
A | Lovastatin | 92.4
| SB 218078 | 46.4
|
7 -
B | Radicicol | 70.3
| Debromohymenialdisine (DBH) | 78.7
|
7 -
C | 17-AAG | 45.3
| Rotenone | 50.3
|
7 -
D | AG1024 | 67.2
| Antimycin A1 | 69.5
|
7 -
E | 1400W, HCl | 86.0
| Leptomycin B* | 32.3
|
7 -
F | AMT, HCl | 93.1
| R59022 | 72.6
|
7 -
G | AG490 | 96.3
| Dioctanoylglycol | 88.2
|
7 -
H | Cucurbitacin I | 64.3
| RHC80267 | 80.1
|
8 -
A | SP600125 | 55.7
| Xanthohumol | 45.6
|
8 -
B | Damnacanthal | 78.8
| C75 | 109.0
|
8 -
C | PD 98059 | 84.0
| Cerulenin | 109.4
|
8 -
D | U0126 | 75.7
| Tunicamycin | 61.9
|
8 -
E | Fumagillin | 92.2
| Deoxynojirimycin | 86.5
|
8 -
F | GM 6001 | 88.5
| Swainsonine | 80.6
|
8 -
G | N-Acetyl-L-cysteine | 98.1
| LY 83583 | 1.7
|
8 -
H | Aminoguanidine, HCl | 90.0
| ODQ | 81.2
|
9 -
A | L-NMMA | 89.0
| Anacardic acid | 75.5
|
9 -
B | PD169316 | 93.1
| Chetomin | 13.6
|
9 -
C | SB 203580 | 81.8
| Dimethyloxalylglycine | 91.2
|
9 -
D | Rapamycin | 70.0
| HR22C16 | 45.4
|
9 -
E | NU1025 | 89.0
| Monastrol | 85.9
|
9 -
F | Benzamide | 91.8
| Nordihydroguaiaretic acid (NDGA) | 86.2
|
9 -
G | D609 | 96.0
| ETYA | 113.3
|
9 -
H | IBMX | 90.3
| Baicalein | 63.1
|
10 -
A | Ro-20-1724 | 93.1
| Nutlin-3 | 65.0
|
10 -
B | Zaprinast | 72.9
| MDM2 inhibitor | 107.9
|
10 -
C | AG1296 | 75.4
| Phenelzine | 82.2
|
10 -
D | LY294002 | 71.5
| Deprenyl | 69.7
|
10 -
E | Wortmannin | 83.5
| Decylubiquinone | 106.8
|
10 -
F | H-89, HCl | 52.8
| Ro 5-4864 | 70.9
|
10 -
G | Bisindolymaleimide I, HCl | 31.5
| Lonidamine | 84.2
|
10 -
H | H-7 | 93.3
| ML-7 | 77.3
|
11 -
A | Staurosporine | 1.7
| Benzylguanine | 82.9
|
11 -
B | cPLA2inhibitor | 85.8
| DFMO | 72.6
|
11 -
C | OBAA | 92.4
| KT 5823 | 106.4
|
11 -
D | Cantharidin | 44.7
| Rp-8-CPT-cGMPS | 88.5
|
11 -
E | Cytostatin | 40.7
| MK 886 | 73.5
|
11 -
F | Cyclosporin A | 54.7
| Clofibrate | 89.5
|
11 -
G | FK-506 | 88.6
| BADGE | 87.8
|
11 -
H | MG-132 | 30.0
| Troglitazone | 75.6
|
12 -
A | Lactacystin | 109.7
| AZT | 94.5
|
12 -
B | Hydroxyurea | 96.8
| Nalidixic acid | 90.9
|
12 -
C | HA1077 | 86.5
| a-Amanitin | 54.9
|
12 -
D | Y27632 | 99.3
| MST-312 | 53.2
|
12 -
E | PP1 (analog) | 79.9
| b-Rubromycin | 77.6
|
12 -
F | PP-H | 96.0
| SB 431542 | 105.6
|
12 -
G | Nocodazole | 48.6
| N1,N12-Diethylspermine (BESpm) | 99.1
|
12 -
H | Dephostatin | 91.3
| Fumonisin B1 | 86.8
|