Well | KIT 1 | KIT 2 | KIT 3 |
compound | 結果 | compound | 結果 | compound | 結果 |
1 -
A | none (DMSO) |
| none (DMSO) |
| none (DMSO) |
|
1 -
B | 5-FU |
| Pifithrin-a (cyclic) |
| ABT-702 |
|
1 -
C | Bestatin Hydrochloride |
| PRIMA-1 |
| Akt Inhibitor IV | Yes
|
1 -
D | Bleomycin sulfate |
| Finasteride |
| Akt Inhibitor VIII, Isozyme-Selective, Akti-1/2 | Yes
|
1 -
E | Cisplatin |
| Aminoglutethimide |
| Akt Inhibitor XI |
|
1 -
F | Methotrexate |
| Formestane |
| compound C |
|
1 -
G | Mitomycin C |
| Mifepristone |
| ATM/ATR kinase inhibitor |
|
1 -
H | Vinblastine sulfate |
| TOFA |
| ATM kinase inhibitor |
|
2 -
A | Paclitaxel |
| Amastatin |
| Aurora kinase/cdk inhibitor |
|
2 -
B | Flutamide |
| Actinonin |
| Aurora kinase inhibitor II |
|
2 -
C | Daunorubicin, HCl |
| Oligomycin |
| Aurora kinase inhibitor III |
|
2 -
D | Doxorubicin, HCl |
| Bafilomycin A1 | Yes
| AG957 |
|
2 -
E | Tamoxifen, citrate |
| HA 14-1 |
| LFM-A13 |
|
2 -
F | Actinomycin D |
| BH3I-1 |
| Terreic acid |
|
2 -
G | Camptothecin |
| LFM-A13 |
| KN-93 |
|
2 -
H | Aclarubicin |
| Terreic acid |
| KN-62 | Yes
|
3 -
A | Etoposide (VP-16) |
| E-64d |
| Lavendustin C |
|
3 -
B | Cytochalasin D |
| ALLN |
| Kenpaullone |
|
3 -
C | 2',5'-dideoxyadenosine |
| CA-074 |
| purvalanol A |
|
3 -
D | AKT inhibitor |
| Pepstatin A |
| Olomoucine |
|
3 -
E | NL-71-101 |
| Z-GLF-CMK |
| Alsterpaullone, 2-cyanoethyl |
|
3 -
F | AG957 |
| RS 102895 |
| Cdk1/2 inhibitor III |
|
3 -
G | KN93 | Yes
| SB 328437 |
| Cdk2/9 inhibitor |
|
3 -
H | Z-VAD-FMK |
| SB 225002 |
| NU6102 |
|
4 -
A | Kenpaullone |
| AMD3100 octahydrochloride |
| Cdk4 inhibitor |
|
4 -
B | Purvalanol A |
| NSC95397 |
| NSC625987 |
|
4 -
C | 3-ATA |
| SC-ααδ9 |
| SB218078 |
|
4 -
D | Olomoucine |
| Amiloride |
| isogranulatimide |
|
4 -
E | TBB |
| Lidocaine |
| Chk2 inhibitor |
|
4 -
F | Sulindac sulfide |
| Monensin |
| Chk2 inhibitor II |
|
4 -
G | Valeryl salicylate |
| Ouabain |
| Ellagic acid (Dihydrate) |
|
4 -
H | NS-398 |
| Sanguinarine | Yes
| TBB |
|
5 -
A | Sodium salicylate |
| Glibenclamide |
| DMAT |
|
5 -
B | Theophylline |
| Dequalinium |
| D4476 |
|
5 -
C | Azacytidine |
| Diazoxide |
| TG003 |
|
5 -
D | Aphidicolin |
| Valinomycin | No
| Diacylglycerol kinase inhibitor II |
|
5 -
E | AG1478 |
| Nigericin |
| IC60211 |
|
5 -
F | Genistein |
| Diltiazem |
| TX-1918 |
|
5 -
G | Manumycin A |
| Nifedipine |
| BPIQ-Ⅱ |
|
5 -
H | FTI-276 |
| Verapamil |
| AG1478 |
|
6 -
A | SU1498 |
| PGP-4008 |
| AG490 |
|
6 -
B | GGTI-286 |
| Fumitremorgin C |
| SU4984 |
|
6 -
C | Dexamethasone |
| A23187 | Yes
| SU5402 |
|
6 -
D | GSK-3 inhibitor II |
| Ionomycin | Yes
| Flt-3 Inhibitor |
|
6 -
E | Scriptaid |
| Thapsigargin | Yes
| cFMS Receptor Tyrosine Kinase Inhibitor |
|
6 -
F | Trichostatin A |
| t-Butylhydroquinone (BHQ) |
| SU6656 |
|
6 -
G | AG825 |
| N-phenylanthranilic acid |
| GSK-3 inhibitor IX | No
|
6 -
H | Cycloheximide |
| DIDS |
| 1-Azakenpaullone |
|
7 -
A | Lovastatin |
| SB 218078 |
| Indirubin-3'-monoxime |
|
7 -
B | Radicicol |
| Debromohymenialdisine (DBH) |
| AG825 |
|
7 -
C | 17-AAG |
| Rotenone |
| AG1024 |
|
7 -
D | AG1024 |
| Antimycin A1 |
| AGL 2263 |
|
7 -
E | 1400W, HCl |
| Leptomycin B* |
| BMS-345541 |
|
7 -
F | AMT, HCl |
| R59022 |
| IKK-2 inhibitor VI |
|
7 -
G | AG490 |
| Dioctanoylglycol |
| IRAK-1/4 inhibitor |
|
7 -
H | Cucurbitacin I | Yes
| RHC80267 |
| JAK Inhibitor I |
|
8 -
A | SP600125 |
| Xanthohumol |
| JAK3 Inhibitor VI |
|
8 -
B | Damnacanthal |
| C75 |
| SP600125 |
|
8 -
C | PD 98059 |
| Cerulenin |
| JNK inhibitor VIII |
|
8 -
D | U0126 |
| Tunicamycin |
| Damnacanthal |
|
8 -
E | Fumagillin |
| Deoxynojirimycin |
| PP2 |
|
8 -
F | GM 6001 |
| Swainsonine |
| ERK inhibitor II |
|
8 -
G | N-Acetyl-L-cysteine |
| LY 83583 | No
| PD98059 | No
|
8 -
H | Aminoguanidine, HCl |
| ODQ |
| U-0126 |
|
9 -
A | L-NMMA |
| Anacardic acid |
| MEK inhibitor I |
|
9 -
B | PD169316 |
| Chetomin | No
| SU11274 |
|
9 -
C | SB 203580 |
| Dimethyloxalylglycine |
| ML-7 |
|
9 -
D | Rapamycin |
| HR22C16 |
| SB202190 |
|
9 -
E | NU1025 |
| Monastrol |
| SB239063 |
|
9 -
F | Benzamide |
| Nordihydroguaiaretic acid (NDGA) |
| AG1296 |
|
9 -
G | D609 |
| ETYA |
| SU11652 | Yes
|
9 -
H | IBMX |
| Baicalein |
| PDGF receptor tyrosine kinase inhibitor V |
|
10 -
A | Ro-20-1724 |
| Nutlin-3 |
| PDGF receptor tyrosine kinase inhibitor IV |
|
10 -
B | Zaprinast |
| MDM2 inhibitor |
| LY-294002 |
|
10 -
C | AG1296 |
| Phenelzine |
| Wortmannin |
|
10 -
D | LY294002 |
| Deprenyl |
| H-89 |
|
10 -
E | Wortmannin | No
| Decylubiquinone |
| 4-cyano-3-methylisoquinoline |
|
10 -
F | H-89, HCl |
| Ro 5-4864 |
| Bisindolymaleimide I, HCl |
|
10 -
G | Bisindolymaleimide I, HCl |
| Lonidamine |
| Go7874 |
|
10 -
H | H-7 |
| ML-7 |
| Rp-8-CPT-cGMPS |
|
11 -
A | Staurosporine | Yes
| Benzylguanine |
| KT5823 |
|
11 -
B | cPLA2inhibitor | Yes
| DFMO |
| PKR inhibitor |
|
11 -
C | OBAA |
| KT 5823 |
| RAF1 kinase inhibitor I |
|
11 -
D | Cantharidin | Yes
| Rp-8-CPT-cGMPS |
| ZM 336372 |
|
11 -
E | Cytostatin |
| MK 886 |
| H-1152 |
|
11 -
F | Cyclosporin A |
| Clofibrate |
| Y-27632 |
|
11 -
G | FK-506 |
| BADGE |
| radicicol |
|
11 -
H | MG-132 | Yes
| Troglitazone |
| PP1 analog |
|
12 -
A | Lactacystin | Yes
| AZT |
| Syk inhibitor |
|
12 -
B | Hydroxyurea |
| Nalidixic acid |
| SB431542 |
|
12 -
C | HA1077 |
| a-Amanitin |
| TGF-b RI kinase inhibitor II |
|
12 -
D | Y27632 |
| MST-312 |
| Tpl2 kinase inhibitor |
|
12 -
E | PP1 (analog) |
| b-Rubromycin |
| TrkA inhibitor |
|
12 -
F | PP-H |
| SB 431542 |
| VEGFR receptor tyrosine kinase inhibitor II |
|
12 -
G | Nocodazole |
| N1,N12-Diethylspermine (BESpm) |
| VEGF recptor 2 kinase inhibitor I |
|
12 -
H | Dephostatin |
| Fumonisin B1 |
| SU1498 |
|